简介 :Sonolisib (PX-866), an improved Wortmannin analogue, is an oral, irreversible, and pan-isoform inhibitor of PI3K (IC50=0.1 nM (p110α), 1.0 nM (p120γ), 2.9 nM (p110δ)). Antitumor activity.
Catalog_No:HY-N6775
Alternative_Names:PX-866
产品一级分类:信号通路
二级分类:生命科学试剂
SMILES:O=C1C([C@@](CC2)([H])[C@@]3(C)C2=O)=C([C@H](OC(C)=O)C3)[C@]4(C)C(/C(C(O[C@@H]4COC)=O)=C\N(CC=C)CC=C)=C1O
Pathway:PI3K/Akt/mTOR
Target:PI3K
Research_Area:Cancer
国际站:Sonolisib