简介 :GN44028 is a hypoxia inducible factor (HIF)-1 inhibitor, with an IC50 of 14 nM. GN44028 inhibits hypoxia-induced HIF-1α transcriptional activity without suppressing HIF-1α mRNA expression, HIF-1α protein accumulation, or HIF-1α/HIF-1β heterodimerization.
Catalog_No:HY-110266
Alternative_Names:
产品一级分类:信号通路
二级分类:生命科学试剂
SMILES:C1(NC2=CC=C(OCCO3)C3=C2)=NNC4=C1CC5=CC=CC=C45
Pathway:Metabolic Enzyme/Protease
Target:HIF/HIF Prolyl-Hydroxylase
Research_Area:Cancer
国际站:GN44028